Introduction
- Organophosphates (OPs) are commonly used pesticides.
- Cause: ingestion of pesticide or following treatment for external parasites.
- Action : organophosphates form a temporarily reversible bond with acetylcholine esterase (AChE) and butyrylcholinesterase (pseudocholinesterase), which becomes permanent with time.
- Signs : cholinergic crisis (excessive parasympathetic stimulation, skeletal muscle stimulation and central stimulation) varying with the compound involved and individual susceptibility.
- Treatment : prompt action required if to be successful.
- Prognosis : good if prompt treatment.
Diagnosis
Clinical signs
- Exact pattern of signs - balance between parasympathetic stimulation, skeletal muscular stimulation and CNS stimulation depends on individual compound, individual animal and level of exposure.
Muscarinic signs
- Hypersalivation.
- Hyperlacrimation.
- Frequent urination and defecation.
- Noisy gastrointestinal activity.
- Bradycardia.
- Pupillary constriction.
Nicotinic signs
- Muscle fasciculation.
- Tremor.
- Twitching.
- Spasms, causing stiff gait or rigid stance.
- Eventually weakness and paralysis.
- Anxiety.
- Restlessness/hyperactivity.
- Anorexia.
- Generalized seizures.
- Death from asphyxiation.
Diagnosis
Differential diagnosis
- Carbamate poisoning
. - Amitraz poisoning
. - Pyrethrum
or pyrethroid poisoning
. - Tremorgenic mycotoxin poisoning.
- Partial motor seizures.
- Metaldehyde poisoning
. - Tetanus
. - Idiopathic epilepsy
. - Strychnine poisoning
. - Lead poisoning
. - Hepatic encephalopathy
. - Caffeine or chocolate overdose.
- Other causes of encephalopathies (neoplasia
, inflammation).
Sequelae
Prognosis
- All but the most severe cases will recover with atropine.
- Guarded: if in coma because of wide variation in response to treatment (which depends on individual susceptibility, compound toxicity, dose, time since exposure, route of exposure).
Expected response to treatment
- Parasympathetic signs treated with atropine should be controlled immediately, but they will recur until organophosphate is excreted.
- Skeletal muscle excitation and CNS signs treated with pralidoxime chloride should disappear over 30 minutes following administration.
Reasons for treatment failure
- Highly toxic compound.
- Treatment too late.
Sources
Publications
Refereed papers
- Fikes J D (1990)Toxicology of selected pesticides, drugs, and chemicals - organophosphorus and carbamate insecticides.Vet Clin North Am Small Anim Pract20(2), 353-367.
Other sources of information
- Blodgett D J (2001)Organophosphate and Carbamate InsecticidesInSmall Animal Toxicology.Eds: M E Peterson and P A Talcott. Philadelphia: W B Saunders. ISBN: 0 7216 7826 2.
- Osweiler G D (1995)Toxicology.Philadelphia: Williams and Wilkins. ISBN: 0 6830 6664 1.
Organization(s)
Veterinary Poisons Information Service (VPIS)- Poisons Unit, Avonley Road, London SE14 5ER, UK. Tel: 020-76359195.



